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A Direct, Regioselective and Atom-Economical Synthesis of 3-Aroyl-N-hydroxy-5-nitroindoles by Cycloaddition of 4-Nitronitrosobenzene with Alkynones
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A Direct, Regioselective and Atom-Economical Synthesis of 3-Aroyl-N-hydroxy-5-nitroindoles by Cycloaddition of 4-Nitronitrosobenzene with Alkynones

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Synthesis and anticancer activity of 2,4-disubstituted furo[3,2-b]indole derivatives

Shi-Hong Zhuang1, Yi-Chien Lin, Li-Chen Chou

  • 1Graduate Institute of Pharmaceutical Chemistry, China Medical University, No. 91 Hsueh-Shih Road, Taichung 40402, Taiwan ROC.

European Journal of Medicinal Chemistry
|July 9, 2013
PubMed

Keywords:
A498 renal cancer cellsAnticancer activityFuro[3,2-b]indole derivativesStructure–activity relationships (SARs)

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