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Imidazolium-based warheads strongly influence activity of water-soluble peptidic transglutaminase inhibitors

Eduard Badarau1, Alexandre Mongeot, Russell Collighan

  • 1School of Life and Health Sciences, Aston University, Aston Triangle, Birmingham B4 7ET, UK.

European Journal of Medicinal Chemistry
|July 10, 2013
PubMed

Keywords:
Coagulation factor XIIIa (FXIIIa)DialkylsulfoniumImidazolium warheadsPeptidic inhibitorsTissue transglutaminase (TG2)

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