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Updated: May 9, 2026

A Fluorescent Screening Assay for Identifying Modulators of GIRK Channels
05:31

A Fluorescent Screening Assay for Identifying Modulators of GIRK Channels

Published on: April 24, 2012

Discovery of 'molecular switches' within a GIRK activator scaffold that afford selective GIRK inhibitors

Wandong Wen1, Wenjun Wu, Ian M Romaine

  • 1College of Science, Northwest Agriculture & Forestry University, Yangling, Shaanxi 712100, China.

Bioorganic & Medicinal Chemistry Letters
|July 11, 2013
PubMed

Keywords:
ActivatorsGIRKInhibitorsK(ir)3.xThallium flux

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