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Identification of potent, selective, CNS-targeted inverse agonists of the ghrelin receptor

Kim F McClure1, Margaret Jackson, Kimberly O Cameron

  • 1Departments of Medicinal Chemistry, Discovery Biology, Drug Metabolism and Pharmaceutical Sciences, Pfizer Worldwide Research and Development, Groton, CT 06340, United States. kim.f.mcclure@pfizer.com

Bioorganic & Medicinal Chemistry Letters
|August 20, 2013
PubMed

Keywords:
AntagonistGhrelinInverse agonistMuscarinicReceptorReceptor occupancy

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