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High-throughput Screening for Small-molecule Modulators of Inward Rectifier Potassium Channels
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High-throughput Screening for Small-molecule Modulators of Inward Rectifier Potassium Channels

Published on: January 27, 2013

Design and bio-evaluation of indole derivatives as potent Kv1.5 inhibitors

Xiaoke Guo1, Qian Yang, Jing Xu

  • 1Jiang Su Key Laboratory of Drug Design and Optimization, China Pharmaceutical University, Nanjing 210009, China; State Key Laboratory of Natural Medicines, China Pharmaceutical University, Nanjing 210009, China.

Bioorganic & Medicinal Chemistry
|September 28, 2013
PubMed

Keywords:
Atrial fibrillation (AF)Indole derivativesKv1.5Structure–activity relationship (SAR)

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