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Updated: May 6, 2026

BRET-based G Protein Biosensors for Measuring G Protein-Coupled Receptor Activity in Live Cells
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Recent development of CB2 selective and peripheral CB1/CB2 cannabinoid receptor ligands

Tapio Nevalainen1

  • 1School of Pharmacy, Faculty of Health Sciences, University of Eastern Finland, Kuopio, P.O. Box 1627, FI-70211 Kuopio, Finland. tapio.nevalainen@uef.fi.

Current Medicinal Chemistry
|October 30, 2013
PubMed
Summary

Selective CB2 receptor ligands offer therapeutic benefits for pain and cancer, minimizing central nervous system side-effects. Recent advancements focus on developing novel CB2 agonists for potential clinical applications.

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