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A Direct, Regioselective and Atom-Economical Synthesis of 3-Aroyl-N-hydroxy-5-nitroindoles by Cycloaddition of 4-Nitronitrosobenzene with Alkynones

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Synthesis and pharmacological evaluation of novel bisindolylalkanes analogues

Ya-Li Song1, Yun-Fang Dong, Tao Yang

  • 1Key Laboratory for Pharmaceutical Quality Control of Hebei Province, College of Pharmaceutical Sciences, Hebei University, Wusi East Road No. 180, Baoding, Hebei 071002, China; Key Laboratory of Medical Chemistry and Molecular Diagnosis, Ministry of Education, Wusi East Road No. 180, Baoding, Hebei 071002, China.

Bioorganic & Medicinal Chemistry
|November 23, 2013
PubMed

Keywords:
AnticancerBisindolylalkaneIndoleThiochroman-4-oneTopoisomerase II

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