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CB2 cannabinoid receptor is a novel target for third-generation selective estrogen receptor modulators bazedoxifene

Pritesh Kumar1, Zhao-Hui Song1

  • 1Department of Pharmacology and Toxicology, University of Louisville School of Medicine, Louisville, KY 40292, United States.

Biochemical and Biophysical Research Communications
|November 27, 2013
PubMed

Keywords:
BazedoxifeneCB1CB2Cannabinoid receptorFDAG protein-coupled receptorGPCRHTRFInverse agonistLasofoxifeneSERMSelective estrogen receptor modulatorcannabinoid receptor 1cannabinoid receptor 2food and drug administrationhomogenous time resolved fluorescenceselective estrogen receptor modulator

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