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BRET-based G Protein Biosensors for Measuring G Protein-Coupled Receptor Activity in Live Cells
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BRET-based G Protein Biosensors for Measuring G Protein-Coupled Receptor Activity in Live Cells

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Insights into the structure of class B GPCRs

Kaspar Hollenstein1, Chris de Graaf2, Andrea Bortolato1

  • 1Heptares Therapeutics Ltd, BioPark, Broadwater Road, Welwyn Garden City, AL7 3AX, UK.

Trends in Pharmacological Sciences
|December 24, 2013
PubMed

Keywords:
class B G protein-coupled receptor (GPCR)corticotropin-releasing factor receptor 1 (CRF(1))crystal structureglucagon receptor (GCGR)ligand binding

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