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Thiazolopyridone ureas as DNA gyrase B inhibitors: optimization of antitubercular activity and efficacy

Ramesh R Kale1, Manoj G Kale1, David Waterson1

  • 1Department of Medicinal Chemistry, AstraZeneca India Pvt. Ltd, Bellary Road, Hebbal, Bangalore 560024, India.

Bioorganic & Medicinal Chemistry Letters
|January 11, 2014
PubMed

Keywords:
DNA gyraseGyrBThiazolopyridone ureasTuberculosis

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