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A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators
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Identification of highly efficacious glucocorticoid receptor agonists with a potential for reduced clinical bone side

Christian Harcken1, Doris Riether, Daniel Kuzmich

  • 1Department of Medicinal Chemistry, Department of Immunology and Inflammation, Department of Chemical Development, Boehringer Ingelheim Pharmaceuticals, Inc. , 900 Ridgebury Road, Ridgefield, Connecticut 06877, United States.

Journal of Medicinal Chemistry
|February 11, 2014
PubMed

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