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In vitro and in vivo biotransformation of WMS-1410, a potent GluN2B selective NMDA receptor antagonist

Evamaria Falck1, Frank Begrow1, Eugen J Verspohl1

  • 1Institut für Pharmazeutische und Medizinische Chemie, Westfälische Wilhelms-Universität, Münster, Germany.

Journal of Pharmaceutical and Biomedical Analysis
|February 19, 2014
PubMed

Keywords:
GluN2B receptor antagonistsIn vitro and in vivo biotransformationLC–MSNMDA receptorRate of degradation

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