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Updated: May 2, 2026

A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators
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A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators

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Unifying family A GPCR theories of activation

Benjamin G Tehan1, Andrea Bortolato1, Frank E Blaney1

  • 1Heptares Therapeutics BioPark, Broadwater Road, Welwyn Garden City AL7 3AX United Kingdom.

Pharmacology & Therapeutics
|February 25, 2014
PubMed

Keywords:
ActivationConservational analysisConstitutive activityGPCR

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