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Updated: May 1, 2026

A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators
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Discovery of substituted benzamides as follicle stimulating hormone receptor allosteric modulators

Henry N Yu1, Thomas E Richardson2, Selva Nataraja3

  • 1EMD Serono Research Institute, 45A Middlesex Turnpike, Billerica, MA 01821, United States; TocopheRx, Inc., Suite 1077, 15 New England Executive Park, Burlington, MA 01803, United States.

Bioorganic & Medicinal Chemistry Letters
|April 2, 2014
PubMed

Keywords:
AgonistAntagonistGPCRGlycoprotein hormoneGonadotropinInfertilityOvaryPAMReproductive

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