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Benzylpiperidine variations on histamine H3 receptor ligands for improved drug-likeness

Kerstin Wingen1, J Stephan Schwed2, Kathleen Isensee1

  • 1Johann Wolfgang Goethe University, Institute of Pharmaceutical Chemistry, Biozentrum, Max-von-Laue-Str. 9, 60438 Frankfurt/Main, Germany.

Bioorganic & Medicinal Chemistry Letters
|April 22, 2014
PubMed

Keywords:
AntagonistsDrug-likenessGPCRHistamine H(3) receptorLipophilicity

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