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Base substituted 5'-O-(N-isoleucyl)sulfamoyl nucleoside analogues as potential antibacterial agents

Bharat Gadakh1, Gaston Vondenhoff1, Eveline Lescrinier1

  • 1KU Leuven, Medicinal Chemistry, Rega Institute for Medical Research, Leuven, Belgium.

Bioorganic & Medicinal Chemistry
|April 22, 2014
PubMed

Keywords:
Aminoacyl-tRNA synthetasesBase modificationsEnzyme inhibitorsIn vitro affinityMolecular modelingNucleoside antibiotics

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