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The discovery of diazepinone-based 5-HT3 receptor partial agonists

David D Manning1, Cheng Guo1, Zhenjun Zhang1

  • 1Albany Molecular Research Inc. (AMRI), 26 Corporate Circle, Albany, NY 12212-5098, United States.

Bioorganic & Medicinal Chemistry Letters
|April 24, 2014
PubMed

Keywords:
5-HT(3) receptor partial agonistAlosetronDiazepinoneIrritable bowel syndrome (IBS)Ligand-gated ion channelRamosetron

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