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Discovery of novel diarylpyrimidines as potent HIV NNRTIs via a structure-guided core-refining approach

Xiao Li1, Wenmin Chen1, Ye Tian1

  • 1Department of Medicinal Chemistry, Key Laboratory of Chemical Biology (Ministry of Education), School of Pharmaceutical Sciences, Shandong University, 44 West Culture Road, 250012 Jinan, Shandong, PR China.

European Journal of Medicinal Chemistry
|April 29, 2014
PubMed

Keywords:
Anti-HIV activitiesDAPYHIV-1HIV-2Molecular modelingStructure–activity relationships

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