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Updated: Apr 29, 2026

Methods for the Discovery of Novel Compounds Modulating a Gamma-Aminobutyric Acid Receptor Type A Neurotransmission
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Discovery of 3-aryl-3-ethoxypropanoic acids as orally active GPR40 agonists

Rieko Takano1, Masao Yoshida1, Masahiro Inoue1

  • 1R&D Division, Daiichi Sankyo Co., Ltd., 1-2-58 Hiromachi, Shinagawa-ku, Tokyo 140-8710, Japan.

Bioorganic & Medicinal Chemistry Letters
|May 20, 2014
PubMed

Keywords:
AgonistDiabetesGPR40Glucose loweringInsulin secretagogue

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