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Updated: Apr 28, 2026

Measuring G-protein-coupled Receptor Signaling via Radio-labeled GTP Binding
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Measuring G-protein-coupled Receptor Signaling via Radio-labeled GTP Binding

Published on: June 9, 2017

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Biased ligands at G-protein-coupled receptors: promise and progress

Jonathan D Violin1, Aimee L Crombie1, David G Soergel1

  • 1Trevena Inc., 1018 West 8th Avenue, Suite A, King of Prussia, PA 19406, USA.

Trends in Pharmacological Sciences
|June 1, 2014
PubMed

Keywords:
TRV027TRV130angiotensinfunctional selectivityopioidβ-arrestin

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