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Methods for the Discovery of Novel Compounds Modulating a Gamma-Aminobutyric Acid Receptor Type A Neurotransmission
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Discovery of WAY-260022, a Potent and Selective Inhibitor of the Norepinephrine Transporter

Lori K Gavrin1, Paige E Mahaney2, Douglas Jenkins2

  • 1Worldwide Medicinal Chemistry, Pfizer Global Research and Development, 200 Cambridge Park Drive, Cambridge, Massachusetts 02140.

ACS Medicinal Chemistry Letters
|June 6, 2014
PubMed

Keywords:
WAY-260022brain penetration, vasomotor symptomsdopamine transporternorepinephrine reuptake inhibitorserotonin transporter

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