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Author Spotlight: Advancing Cellular and Protein Engineering to Control Biological Functions and Develop Novel Therapies
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Discovery of LAS101057: A Potent, Selective, and Orally Efficacious A2B Adenosine Receptor Antagonist

Paul Eastwood1, Cristina Esteve1, Jacob González1

  • 1Almirall, R&D Centre, Ctra. Laureà Miró 408, 08980-Sant Feliu de Llobregat, Barcelona, Spain.

ACS Medicinal Chemistry Letters
|June 6, 2014
PubMed

Keywords:
A2B adenosine receptor antagonistclinical candidateovalbumin mouse model

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