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A Pipeline to Investigate the Structures and Signaling Pathways of Sphingosine 1-Phosphate Receptors
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Discovery of CS-0777: A Potent, Selective, and Orally Active S1P1 Agonist

Takahide Nishi1, Shojiro Miyazaki1, Toshiyasu Takemoto1

  • 1Lead Discovery & Optimization Research Laboratories I, Cardiovascular-Metabolics Research Laboratories, and Drug Metabolism & Pharmacokinetics Research Laboratories, Daiichi Sankyo Co., Ltd. , 1-2-58 Hiromachi, Shinagawa-ku, Tokyo, 140-8710, Japan.

ACS Medicinal Chemistry Letters
|June 6, 2014
PubMed

Keywords:
CS-0777EAEMSS1P1agonistlymphocyte

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