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Identification of Novel CK2 Kinase Substrates Using a Versatile Biochemical Approach
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Potent and Selective Inhibitors of CK2 Kinase Identified through Structure-Guided Hybridization

James E Dowling1, Claudio Chuaqui1, Timothy W Pontz1

  • 1AstraZeneca , Oncology Innovative Medicines Unit, 35 Gatehouse Drive, Waltham, Massachusetts 02145, United States.

ACS Medicinal Chemistry Letters
|June 6, 2014
PubMed

Keywords:
CK2casein kinasepyrazolo[1,5-a]pyrimidinestructure-based design

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