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Identification of Tetrahydropyrido[4,3-d]pyrimidine Amides as a New Class of Orally Bioavailable TGR5 Agonists

David W Piotrowski1, Kentaro Futatsugi1, Joseph S Warmus1

  • 1Pfizer Worldwide Research and Development , Groton, Connecticut 06340, United States.

ACS Medicinal Chemistry Letters
|June 6, 2014
PubMed

Keywords:
GLP-1GPCRTGR5agonistdiabetes

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