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Probing the Binding Site of Bile Acids in TGR5

Antonio Macchiarulo1, Antimo Gioiello1, Charles Thomas2

  • 1Dipartimento di Chimica e Tecnologia del Farmaco, Università degli Studi di Perugia , 06123 Perugia, Italy.

ACS Medicinal Chemistry Letters
|June 6, 2014
PubMed

Keywords:
Bile acidsGPCRTGR5diabeteshomology modelingmolecular dockingsite-directed mutagenesis

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