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Potent DGAT1 Inhibitors in the Benzimidazole Class with a Pyridyl-oxy-cyclohexanecarboxylic Acid Moiety

Shuwen He1, Qingmei Hong1, Zhong Lai1

  • 1Discovery and Preclinical Sciences, Merck Research Laboratories , 2000 Galloping Hill Road, Kenilworth, New Jersey 07033, United States.

ACS Medicinal Chemistry Letters
|June 6, 2014
PubMed

Keywords:
ACAT1DGAT1benzimidazolecyclohexanecarboxylic acidepimerizationinhibitorlipid tolerance testmetabolite

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