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Aminopyrazole-Phenylalanine Based GPR142 Agonists: Discovery of Tool Compound and in Vivo Efficacy Studies

Ming Yu1, Mike Lizarzaburu1, Alykhan Motani1

  • 1Amgen Inc. , 1120 Veterans Boulevard, South San Francisco, California 94080, United States.

ACS Medicinal Chemistry Letters
|June 6, 2014
PubMed

Keywords:
GPR142 agonistaminopyrazole−phenylalaninehuman islet transplantinsulin secretagogueoral glucose tolerance testprodrugtype 2 diabetes

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