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Updated: Apr 28, 2026

15N CPMG Relaxation Dispersion for the Investigation of Protein Conformational Dynamics on the µs-ms Timescale
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Optimizing the Physicochemical Properties of Raf/MEK Inhibitors by Nitrogen Scanning

Toshihiro Aoki1, Ikumi Hyohdoh1, Noriyuki Furuichi1

  • 1Research Division, Chugai Pharmaceutical Co., Ltd. , 200 Kajiwara, Kamakura, Kanagawa 247-8530, Japan.

ACS Medicinal Chemistry Letters
|June 6, 2014
PubMed

Keywords:
CH5126766MEKNitrogen scanRO5126766Rafkinase inhibitor

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