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Structure-Guided Rescaffolding of Selective Antagonists of BCL-XL

Michael F T Koehler1, Philippe Bergeron1, Edna F Choo1

  • 1Departments of Discovery Chemistry, Drug Metabolism and Pharmacokinetics, and Early Discovery Biochemistry, Genentech, Inc. , 1 DNA Way, South San Francisco, California 94080, United States.

ACS Medicinal Chemistry Letters
|June 20, 2014
PubMed

Keywords:
BCL-2BCL-XLapoptosiscancer

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