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Discovery of highly potent DPP-4 inhibitors by hybrid compound design based on linagliptin and alogliptin

Zeng-Wei Lai1, Chunhong Li1, Jun Liu2

  • 1State Key Laboratory of Natural Medicines and Center of Drug Discovery, China Pharmaceutical University, 24 Tongjia Xiang, Nanjing 210009, PR China.

European Journal of Medicinal Chemistry
|July 5, 2014
PubMed

Keywords:
AlogliptinDPP-4 inhibitorsDiabetesHybrid compound designLinagliptin

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