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The impact of cyclopropane configuration on the biological activity of cyclopropyl-epothilones

Fabienne Z Gaugaz1, Mariano Redondo-Horcajo, Isabel Barasoain

  • 1ETH Zürich, Department of Chemistry & Applied Biosciences, Institute of Pharmaceutical Sciences, HCI H405, Vladimir-Prelog-Weg 4, 8093 Zürich (Switzerland).

Chemmedchem
|July 22, 2014
PubMed

Keywords:
cancerepothilonesinhibitorsmicrotubulesstereoselective synthesisstructure-activity relationships

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