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Optimization of 1,2,4-Triazolopyridines as Inhibitors of Human 11β-Hydroxysteroid Dehydrogenase Type 1 (11β-HSD-1)

Jun Li1, Lawrence J Kennedy1, Haixia Wang1

  • 1Department of Medicinal Chemistry, Department of Biology, Lead Evaluation, CADD, Department of Pharmaceutical Candidate Optimization, Bristol-Myers Squibb , Bldg 13, Princeton, New Jersey 08543-5400, United States.

ACS Medicinal Chemistry Letters
|July 23, 2014
PubMed

Keywords:
Enzyme inhibitorshuman 11β-hydroxysteroid dehydrogenase-type 1triazolopyridines

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