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Updated: Apr 26, 2026

Preparation of Stable Bicyclic Aziridinium Ions and Their Ring-Opening for the Synthesis of Azaheterocycles
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Novel piperazinediones as antitumor agents

Chun-Li Wang1, On Lee2, George Hsiao3

  • 1School of Pharmacy, College of Pharmacy, Taipei Medical University, Taipei, Taiwan, R.O.C.

Anticancer Research
|July 31, 2014
PubMed

Keywords:
COMPARE algorithmDTPNCI-60 anticancer screeningNCI/NIHPiperazinedionesazatyrosinamidein vivo antitumor activitymechanism of action predictiontubulin polymerization inhibitor

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