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"Switch off/switch on" regulation of drug cytotoxicity by conjugation to a cell targeting peptide

Yossi Gilad1, Michael A Firer2, Alex Rozovsky1

  • 1Department of Biological Chemistry, Ariel University, Ariel, 40700, Israel; The Julius Spokojny Bioorganic Chemistry Laboratory, Department of Chemistry, Bar Ilan University, Ramat Gan, 52900, Israel.

European Journal of Medicinal Chemistry
|August 2, 2014
PubMed

Keywords:
Amino acid platformControlled drug releasePeptide–drug conjugatesProdrugSolid phase organic synthesis

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