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Pyridine-3-carboxamide-6-yl-ureas as novel inhibitors of bacterial DNA gyrase: structure based design, synthesis, SAR

Ian A Yule1, Lloyd G Czaplewski2, Stephanie Pommier2

  • 1School of Chemistry, University of Leeds, Leeds LS2 9JT, UK.

European Journal of Medicinal Chemistry
|August 20, 2014
PubMed

Keywords:
Bacterial resistanceDNA gyraseMolecular modellingPyridine-3-carboxamide

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