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Methods for the Discovery of Novel Compounds Modulating a Gamma-Aminobutyric Acid Receptor Type A Neurotransmission
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Conformationally Restricted GABA with Bicyclo[3.1.0]hexane Backbone as the First Highly Selective BGT-1 Inhibitor

Takaaki Kobayashi1, Akihiro Suemasa1, Arisa Igawa1

  • 1Faculty of Pharmaceutical Sciences, Hokkaido University , Kita-12, Nishi-6, Kita-ku, Sapporo 060-0812, Japan.

ACS Medicinal Chemistry Letters
|August 23, 2014
PubMed

Keywords:
BGT-1GABAGATconformational restrictioncyclopropane

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