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Identification of a nonbasic melanin hormone receptor 1 antagonist as an antiobesity clinical candidate

William N Washburn1, Mark Manfredi, Pratik Devasthale

  • 1Metabolic Diseases Chemistry, ‡Metabolic Diseases Biology, §Preclinical Candidate Optimization Metabolism and Pharmacokinetics, ∥Discovery Chemistry Synthesis, ⊥Preclinical Candidate Optimization Discovery Toxicology, #Preclinical Candidate Optimization Discovery Bioanalytical Research, ∞Preclinical Candidate Optimization Biotransformation, ×Preclinical Candidate Optimization Pharmaceutics, and ○Preclinical Candidate Optimization DAS SPS, Research and Development, Bristol-Myers Squibb Co. , Princeton, New Jersey 08543-5400, United States.

Journal of Medicinal Chemistry
|August 29, 2014
PubMed

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