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Assays for Validating Histone Acetyltransferase Inhibitors
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Novel antiproliferative chimeric compounds with marked histone deacetylase inhibitory activity

Elisa Giacomini1, Angela Nebbioso2, Alfonso Ciotta2

  • 1Department of Pharmacy and Biotechnology, University of Bologna , Via Belmeloro 6, 40126 Bologna, Italy ; Department of Drug Discovery and Development, Italian Institute of Technology , Via Morego 30, 16163 Genova, Italy.

ACS Medicinal Chemistry Letters
|September 16, 2014
PubMed

Keywords:
HDAC inhibitionMultifunctional ligandsantiproliferative activitychimeric compoundstilbene

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