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Computational & experimental evaluation of the structure/activity relationship of β-carbolines as DYRK1A inhibitors

Binia Drung1, Christoph Scholz1, Valéria A Barbosa2

  • 1Clemens Schöpf-Institute of Organic Chemistry and Biochemistry, Technische Universität Darmstadt, Alarich-Weiss-Str. 4, 64287 Darmstadt, Germany.

Bioorganic & Medicinal Chemistry Letters
|September 22, 2014
PubMed

Keywords:
DYRK1ADockingInhibitorMAO-APharmacophoreSARβ-Carboline

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