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Metabolic stability optimization and metabolite identification of 2,5-thiophene amide 17β-hydroxysteroid

Emanuele M Gargano1, Enrico Perspicace1, Nina Hanke2

  • 1Pharmaceutical and Medicinal Chemistry, Saarland University, Campus C2(3), D-66123 Saarbrücken, Germany.

European Journal of Medicinal Chemistry
|September 27, 2014
PubMed

Keywords:
17β-HSD2Inhibitor designMetabolic stabilityMetabolite identificationOsteoporosiscLogP

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