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A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators
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G-protein-coupled receptor type A heteromers as an emerging therapeutic target

Diego Guidolin1, Luigi F Agnati, Manuela Marcoli

  • 1University of Padova, Department of Molecular Medicine , via Gabelli 65, 35121 Padova , Italy +39 049 8272316 ; +39 049 8272319 ; diego.guidolin@unipd.it.

Expert Opinion on Therapeutic Targets
|November 11, 2014
PubMed
Abstract

Keywords:
G protein-coupled receptorsallosteric modulationheteromersneurologyneuropsychopharmacologyreceptor-receptor interactions

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