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New trisubstituted 1,2,4-triazoles as ghrelin receptor antagonists

Anne-Laure Blayo1, Mathieu Maingot1, Babette Aicher2

  • 1Institut des Biomolécules Max Mousseron (IBMM), UMR 5247, CNRS-Université Montpellier I et Université Montpellier II, BP 14491, Faculté de Pharmacie, bât. E, 3(ème) étage, 15 avenue Charles Flahault, 34093 Montpellier Cedex 5, France.

Bioorganic & Medicinal Chemistry Letters
|December 2, 2014
PubMed

Keywords:
1,2,4-Triazole scaffoldAntagonistsGHS-R1a, ghrelin receptorSAR studyStructural modulation

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