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Preparation of Stable Bicyclic Aziridinium Ions and Their Ring-Opening for the Synthesis of Azaheterocycles
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Structure-activity relationships (SAR) and structure-kinetic relationships (SKR) of bicyclic heteroaromatic acetic

Juan Antonio Alonso1, Miriam Andrés1, Mónica Bravo1

  • 1Almirall R&D Centre, Laureano Miró, 408-410, 08980 Sant Feliu de Llobregat, Barcelona, Spain.

Bioorganic & Medicinal Chemistry Letters
|December 2, 2014
PubMed

Keywords:
CRTh2 antagonistReceptor residence timeStructure–activity relationship (SAR)Structure–kinetic relationship (SKR)

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