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Access channels to the buried active site control substrate specificity in CYP1A P450 enzymes

Philippe Urban1, Gilles Truan1, Denis Pompon1

  • 1Université de Toulouse, INSA, UPS, INP, LISBP, 135 Avenue de Rangueil, F-31077 Toulouse, France; INRA, UMR792 Ingénierie des Systèmes Biologiques et des Procédés, F-31400 Toulouse, France; CNRS, UMR5504, 135 Avenue de Rangueil, F-31400 Toulouse, France.

Biochimica Et Biophysica Acta
|December 23, 2014
PubMed
Abstract

Keywords:
CAVERCYP1A1ChannelChimeraPolycyclicSelectivity

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