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Potent and selective MAO-B inhibitory activity: amino- versus nitro-3-arylcoumarin derivatives

Maria João Matos1, Fernanda Rodríguez-Enríquez2, Santiago Vilar3

  • 1Departamento de Química Orgánica, Facultad de Farmacia, Universidad de Santiago de Compostela, 15782 Santiago de Compostela, Spain.

Bioorganic & Medicinal Chemistry Letters
|December 24, 2014
PubMed

Keywords:
3-ArylcoumarinsADME theoretical propertiesDocking studiesMonoamine oxidase inhibitorsPAMPA assayPerkin reaction

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