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Updated: Apr 19, 2026

Preparation and In Vivo Use of an Activity-based Probe for N-acylethanolamine Acid Amidase
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Inhibition of Insulin-Regulated Aminopeptidase (IRAP) by Arylsulfonamides

Sanjay R Borhade1, Ulrika Rosenström1, Jonas Sävmarker2

  • 1Organic Pharmaceutical Chemistry, Department of Medicinal Chemistry, BMC, Uppsala University P.O. Box 574, 751 23 Uppsala (Sweden).

Chemistryopen
|January 6, 2015
PubMed

Keywords:
aminopeptidasesarylsulfonamidescognitive enhancersinsulin-regulated aminopeptidase (IRAP)structure–activity relationships

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