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Fluoro-substituted phenylazocarboxamides: Dopaminergic behavior and N-arylating properties for irreversible binding

Amelie L Bartuschat1, Tamara Schellhorn1, Harald Hübner1

  • 1Department of Chemistry and Pharmacy, Friedrich-Alexander-Universität Erlangen-Nürnberg, Schuhstraße 19, 91052 Erlangen, Germany.

Bioorganic & Medicinal Chemistry
|January 8, 2015
PubMed

Keywords:
AzocarboxamideBioisosteresCovalent ligandsD(3) receptorDopamineGPCR

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