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Transport Properties of Ibuprofen Encapsulated in Cyclodextrin Nanosponge Hydrogels: A Proton HR-MAS NMR Spectroscopy Study
Published on: August 15, 2016
[Effect of the microencapsulation process parameters piroxicam by complex coacervation]
L Lamoudi1, J-C Chaumeil2, K Daoud1
1Laboratoire des phénomènes de transfert, faculté de génie mécanique et de génie des procédés, université des sciences et de la technologie Houari Boumediene, BP 32 El Alia, Bab Ezzouar, Alger, Algérie.
This study optimized piroxicam microencapsulation using a gelatin-acacia system, achieving over 70% efficiency. Optimal parameters included a 5:3 gelatin to acacia ratio and 60 minutes crosslinking time for stable microcapsules.
Area of Science:
- Pharmaceutical Sciences
- Materials Science
Background:
- Complex coacervation using a gelatin-acacia system is a method for microencapsulating piroxicam.
- Piroxicam microencapsulation aims to improve drug delivery and stability.
Purpose of the Study:
- To investigate and optimize formulation and process parameters for piroxicam microencapsulation.
- To evaluate the properties of microcapsules produced via complex coacervation.
Main Methods:
- Studied the impact of gelatin/gum acacia ratio, core/wall ratio, crosslinking agent concentration, and crosslinking time.
- Evaluated microcapsule properties including shape, coacervation efficiency, diameter, and stability.
Main Results:
- Microcapsules exhibited a spherical shape with coacervation efficiency exceeding 70% and average diameters below 250 microns.
- Optimal conditions were identified as a 5:3 gelatin/acacia ratio, 1:4 core/wall ratio, 2 mL crosslinking agent, and 60 minutes crosslinking time.
- The resulting microcapsules demonstrated good stability.
Conclusions:
- The gelatin-acacia complex coacervation system is effective for piroxicam microencapsulation.
- Specific formulation and process parameters significantly influence microcapsule characteristics and efficiency.
- Optimized microcapsules offer a promising approach for piroxicam delivery systems.
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