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Structure-Based Drug Design of Novel, Potent, and Selective Azabenzimidazoles (ABI) as ATR Inhibitors

Paul A Barsanti1, Yue Pan1, Yipin Lu1

  • 1Global Discovery Chemistry/Oncology, Novartis Institutes for Biomedical Research , 5300 Chiron Way, Emeryville, California 94608, United States.

ACS Medicinal Chemistry Letters
|January 16, 2015
PubMed

Keywords:
ATRCYP3A4 TDIaldehyde oxidasestructure-based drug design

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